InChi: InChI=1S/C40H37N5O/c1-3-11-29(12-4-1)27-44-36-17-9-7-15-34(36)42-39(44)32-19-21-33(22-20-32)46-28-38(30-23-25-41-26-24-30)45-37-18-10-8-16-35(37)43-40(45)31-13-5-2-6-14-31/h1-22
9 μM and the Vmax value is 3
but it has different pharmacological properties than typical TCAs as recent research suggests that tianeptine produces its antidepressant effects through indirect alteration of glutamate receptor activity (i
5H-cyclopenta[c]isochromene-1-carboxylic acid
Solubility: H2O : 25 mg/mL (6
JKC363 TFA Catalog No.:M17673-C InChi: InChI=1S/C40H37N5O/c1-3-11-29(12-4-1)27-44-36-17-9-7-15-34(36)42-39(44)32-19-21-33(22-20-32)46-28-38(30-23-25-41-26-24-30)45-37-18-10-8-16-35(37)43-40(45)31-13-5-2-6-14-31/h1-22JKC363 TFA, a selective melanocortin MC4 receptor antagonist, has a 90 fold higher affinity at the MC4 receptor (IC50=0. 5 nM) than at the MC3 receptor (44. 9 nM). JKC363 TFA blocks the stimulatory effect of MSH on TRH release. Anti hyperalgesic effect. Product information Molecular Weight: 1620. 73 Formula: C71H92F3N19O18S2 Chemical Name: (S) 3 ((S) 2 ((S) 1 (((4R, 10S, 13S, 16R, 19S, 22S, 25S) 19 ((1H imidazol 4 yl)methyl) 10 ((1H indol 3 yl)methyl)
